| Ident. | Authors (with country if any) | Title |
|---|
| 004408 (2006) |
Syaulan Yang [Taïwan] ; Shu-Jen Chen [Taïwan] ; Min-Feng Hsu [Taïwan] ; Jen-Dar Wu [Taïwan] ; Chien-Te K. Tseng [États-Unis] ; Yu-Fan Liu [Taïwan] ; Hua-Chien Chen [Taïwan] ; Chun-Wei Kuo [Taïwan] ; Chi-Shen Wu [Taïwan] ; Li-Wen Chang [Taïwan] ; Wen-Chang Chen [Taïwan] ; Shao-Ying Liao [Taïwan] ; Teng-Yuan Chang [Taïwan] ; Hsin-Hui Hung [Taïwan] ; Hui-Lin Shr [Taïwan] ; Cheng-Yuan Liu [Taïwan] ; Yu-An Huang [Taïwan] ; Ling-Yin Chang [Taïwan] ; Jen-Chi Hsu [Taïwan] ; Clarence J. Peters [États-Unis] ; Andrew H.-J. Wang [Taïwan] ; Ming-Chu Hsu [Taïwan] | Synthesis, crystal structure, structure-activity relationships, and antiviral activity of a potent SARS coronavirus 3CL protease inhibitor |
| 004421 (2006) |
Kuo-Chen Chou [États-Unis, République populaire de Chine] ; Dong-Qing Wei [États-Unis, République populaire de Chine] ; Qi-Shi Du [États-Unis, République populaire de Chine] ; Suzanne Sirois [États-Unis, Canada] ; Wei-Zhu Zhong [États-Unis] | Progress in computational approach to drug development against SARS |
| 004428 (2006) |
Roberto Di Santo [Italie] ; Roberta Costi [Italie] ; Alessandra Roux [Italie] ; Marino Artico [Italie] ; Antonio Lavecchia [Italie] ; Luciana Marinelli [Italie] ; Ettore Novellino [Italie] ; Lucia Palmisano [Italie] ; Mauro Andreotti [Italie] ; Roberta Amici [Italie] ; Clementina Maria Galluzzo [Italie] ; Lucia Nencioni [Italie] ; Anna Teresa Palamara [Italie] ; Yves Pommier [États-Unis] ; Christophe Marchand [États-Unis] | Novel bifunctional quinolonyl diketo acid derivatives as HIV-1 integrase inhibitors : Design, synthesis, biological activities, and mechanism of action |
| 004451 (2006) |
Andrea J. Dooley [États-Unis] ; Nice Shindo [États-Unis] ; Barbara Taggart [États-Unis] ; Jewn-Giew Park [États-Unis] ; Yuan-Ping Pang [États-Unis] | From genome to drug lead : Identification of a small-molecule inhibitor of the SARS virus |
| 004472 (2006) |
LILI CHEN [République populaire de Chine] ; JIAN LI [République populaire de Chine] ; CHENG LUO [République populaire de Chine] ; HONG LIU [République populaire de Chine] ; WEIJUN XU [Singapour] ; GANG CHEN [Singapour] ; OI WAH LIEW [Singapour] ; WEILIANG ZHU [République populaire de Chine] ; CHUM MOK PUAH [Singapour] ; XU SHEN [République populaire de Chine] ; HUALIANG JIANG [République populaire de Chine] | Binding interaction of quercetin -3 -β -galactoside and its synthetic derivatives with SARS-CoV 3CLpro : Structure-activity relationship studies reveal salient pharmacophore features |
| 004A02 (2005) |
Arun K. Ghosh [Géorgie (pays), États-Unis] ; Kai Xi [Géorgie (pays), États-Unis] ; Kiira Ratia [Géorgie (pays)] ; Bernard D. Santarsiero [Géorgie (pays)] ; Wentao Fu [Géorgie (pays)] ; Brian H. Harcourt [Géorgie (pays)] ; Paul A. Rota [Géorgie (pays)] ; Susan C. Baker [Géorgie (pays)] ; Michael E. Johnson [Géorgie (pays)] ; Andrew D. Mesecar [Géorgie (pays)] | Design and Synthesis of Peptidomimetic Severe Acute Respiratory Syndrome Chymotrypsin-like Protease Inhibitors |
| 004A17 (2005) |
Ulrich Kaeppler [Allemagne] ; Nikolaus Stiefl [Allemagne] ; Markus Schiller [Allemagne] ; Radim Vicik [Allemagne] ; Alexander Breuning [Allemagne] ; Werner Schmitz [Allemagne] ; Daniel Rupprecht [Allemagne] ; Carsten Schmuck [Allemagne] ; Knut Baumann [Allemagne] ; John Ziebuhr [Allemagne] ; Tanja Schirmeister [Allemagne] | A New Lead for Nonpeptidic Active-Site-Directed Inhibitors of the Severe Acute Respiratory Syndrome Coronavirus Main Protease Discovered by a Combination of Screening and Docking Methods‖ |
| 004D51 (2005) |
Li-Rung Chen [Taïwan] ; Yu-Chin Wang [Taïwan] ; YI WEN LIN [Taïwan] ; Shan-Yen Chou [Taïwan] ; Shyh-Fong Chen [Taïwan] ; LEE TAI LIU [Taïwan] ; Ying-Ta Wu [Taïwan] ; Chih-Jung Kuo [Taïwan] ; Tom Shieh-Shung Chen [Taïwan] ; Shin-Hun Juang [Taïwan] | Synthesis and evaluation of isatin derivatives as effective SARS coronavirus 3CL protease inhibitors |
| 004D70 (2005) |
Erika Martina [Allemagne] ; Nikolaus Stiefl [Allemagne] ; Björn Degel [Allemagne] ; Franziska Schulz [Allemagne] ; Alexander Breuning [Allemagne] ; Markus Schiller [Allemagne] ; Radim Vicik [Allemagne] ; Knut Baumann [Allemagne] ; John Ziebuhr [Allemagne] ; Tanja Schirmeister [Allemagne] | Screening of electrophilic compounds yields an aziridinyl peptide as new active-site directed SARS-CoV main protease inhibitor |
| 004E04 (2005) |
Jiun-Jie Shie [Taïwan] ; Jim-Min Fang [Taïwan] ; Tun-Hsun Kuo [Taïwan] ; Chih-Jung Kuo [Taïwan] ; Po-Huang Liang [Taïwan] ; Hung-Jyun Huang [Taïwan] ; Yin-Ta Wu [Taïwan] ; Jia-Tsrong Jan [Taïwan] ; Yih-Shyun E. Cheng [Taïwan] ; Chi-Huey Wong [Taïwan] | Inhibition of the severe acute respiratory syndrome 3CL protease by peptidomimetic α,β-unsaturated esters |
| 005525 (2004) |
Jeffrey H. Toney [États-Unis] ; Sonia Navas-Martín [États-Unis] ; Susan R. Weiss [États-Unis] ; Andreas Koeller [États-Unis] | Sabadinine: A Potential Non-Peptide Anti-Severe Acute-Respiratory-Syndrome Agent Identified Using Structure-Aided Design |
| 005A58 (2004) |
Rajendra P. Jain [Canada] ; Hanna I. Pettersson ; JIANMIN ZHANG ; Katherine D. Aull ; Pascal D. Fortin ; Carly Huitema ; Lindsay D. Eltis ; Jonathan C. Parrish ; Michael N. G. James ; David S. Wishart ; John C. Vederas | Synthesis and evaluation of keto-glutamine analogues as potent inhibitors of severe acute respiratory syndrome 3CLpro |
| 005A83 (2004) |
Mayuko Takeda-Shitaka [Japon] ; Daisuke Takaya [Japon] ; Chieko Chiba [Japon] ; Hirokazu Tanaka [Japon] ; Hideaki Umeyama [Japon] | Protein Structure Prediction in Structure based drug design : Protein structure prediction in medicinal chemistry |
| 006392 (2003) |
Ekachai Jenwitheesuk [États-Unis] ; Ram Samudrala [États-Unis] | Identifying inhibitors of the SARS coronavirus proteinase |
| 006409 (2003) |
Angelo Ranise [Italie] ; Andrea Spallarossa [Italie] ; Silvia Schenone [Italie] ; Olga Bruno [Italie] ; Francesco Bondavalli [Italie] ; Laura Vargiu [Italie] ; Tiziana Marceddu [Italie] ; Massimo Mura [Italie] ; Paolo La Colla [Italie] ; Alessandra Pani [Italie] | Design, synthesis, SAR, and molecular modeling studies of acylthiocarbamates: A novel series of potent non-nucleoside HIV-1 reverse transcriptase inhibitors structurally related to phenethylthiazolylthiourea derivatives |
| 006513 (1998) |
M. Artico [Italie] ; R. Di Santo [Italie] ; R. Costi [Italie] ; E. Novellino [Italie] ; G. Greco [Italie] ; S. Massa [Italie] ; E. Tramontano [Italie] ; M. E. Marongiu [Italie] ; A. De Montis [Italie] ; P. La Colla [Italie] | Geometrically and conformationally restrained cinnamoyl compounds as inhibitors of HIV-1 integrase : Synthesis, biological evaluation, and molecular modeling |
